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Peptide Blend • 2-Component Formulation

Wolverine BPC-157 / TB-500

Two repair-associated peptides co-formulated in one 20 mg vial at a 1:1 ratio. Sold for tendon, ligament and soft-tissue recovery. No study has ever tested the combination, and no published human study establishes a subcutaneous amount for either component on its own.

Overview

Wolverine is a vendor name for a pre-mixed vial containing two synthetic peptides, BPC-157 and TB-500, supplied together as a single lyophilised powder. Athena lists it at 20 mg per vial, 10 mg of each, which is a 1:1 ratio. It is marketed for tendon, ligament and soft-tissue recovery, and the name is a marketing name rather than a compound name — there is no substance called "Wolverine."

ComponentAmountWhat it isProposed role in the blend
BPC-157 (Body Protection Compound)10 mgSynthetic 15-amino-acid partial sequence of a protein found in human gastric juiceAngiogenesis and nitric oxide signalling; connective-tissue and gastrointestinal repair
TB-500 (Thymosin Beta-4 Fragment)10 mgSynthetic 7-amino-acid fragment (Ac-LKKTETQ) of the 43-amino-acid protein thymosin beta-4Actin sequestration, cell migration and tissue remodelling

What the fixed ratio means in practice

Because both peptides sit in one vial, a draw delivers them in the proportion the vial was filled at and no other. A 0.5 mg draw is 0.25 mg of BPC-157 and 0.25 mg of TB-500. Neither can be increased, reduced or stopped without doing the same to the other, which is the main practical difference between this vial and the two compounds bought separately. The individual profiles for BPC-157 and TB-500 set out what is known about each on its own.

What the evidence does and does not cover

The rationale for pairing them is that they are associated with different repair mechanisms — vascular and cytoprotective on one side, cytoskeletal and migratory on the other — so combining them might do more than either alone. That rationale is plausible and it is also entirely untested. No published study examines these two peptides in combination, in any model system. The word "synergy" is a specific pharmacological claim requiring experimental validation, and none exists here.

The component evidence is thinner than the marketing implies. Both peptides have a substantial preclinical literature, almost all of it in rodents. Neither has a published human study establishing a subcutaneous amount, schedule or duration; the handful of human BPC-157 reports used intravenous, intra-articular and intravesical routes, and the human thymosin beta-4 work used the full protein rather than the TB-500 fragment. Both are classified by the FDA as Category 2 bulk drug substances — identified as presenting significant safety risks and prohibited from compounding for human use.

Dosage & Reconstitution

Vial strength
20 mg
BAC water added
3 mL
Final concentration
~6.67 mg/mL
WeeksDosageSyringe units (U-100)
Weeks 1–20.25 mg3.75 units0.04 mL
Weeks 3–80.5 mg7.5 units0.07 mL

FrequencyOnce daily, subcutaneous, as a four-to-eight-week course followed by a break.

Note

For review — no human dosing exists for this blend. Wolverine has never been studied as a combination, so there is no established amount and no established frequency; the two rows in the chart are the amounts circulated for it, given as the total the vial delivers. The concentration strip above the chart is calculated from the vial and water volume and is correct.

Unverified — no study of the blend establishes a course length or a frequency, and no published human study establishes a subcutaneous schedule for either component on its own.

The amount charted is the total the vial delivers, not a figure for either peptide on its own. Athena lists the vial as 10 mg of BPC-157 and 10 mg of TB-500 — 20 mg in total at a 1:1 ratio — so a 0.5 mg draw carries 0.25 mg of each, in a proportion fixed by the vial rather than chosen. The two rows are the two amounts circulated for this blend, 250 mcg and 500 mcg of total blend daily; this page puts the lower one first because starting low is the conservative reading, not because a study sequenced them that way. Neither figure comes from a trial, and the four-to-eight-week course is the circulated structure rather than a finding. Made up with 3 mL the vial is about 6.7 mg/mL, which puts the two rows at 3.75 and 7.5 units — both small draws, well inside a 50-unit syringe. One practical consequence: at these amounts a single 20 mg vial holds forty to eighty daily doses, far more than the roughly four weeks a reconstituted vial keeps for under refrigeration, so most of a vial made up all at once is not usable. Because the two peptides are fixed in one vial they cannot be titrated separately the way each was studied on its own.

What this evidence establishes. No human dosing exists for the Wolverine blend. It has never been studied as a combination — there is no trial of the blend, no validated ratio and no established frequency. Nor does the component literature supply one: no published human study establishes a subcutaneous amount, schedule or duration for BPC-157 or for TB-500, and the handful of human reports that exist for BPC-157 used other routes. Because a blend is supplied at a fixed ratio in a single vial, the amount of each component is set by the vial rather than chosen.

For educational and laboratory research purposes only. It does not provide medical advice, dosing recommendations, or instructions for human or veterinary use. Syringe units assume a U-100 syringe, on which 1 mL is 100 units and a 50-unit syringe holds 0.5 mL.

Component Mechanisms

These mechanisms come from preclinical research on the individual peptides. None of it was generated with the two co-administered.

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BPC-157: Angiogenesis and NO

Modulates the nitric oxide system and promotes blood-vessel formation; protects gastrointestinal mucosa. Rodent models of tendon, ligament and gut injury. FDA Category 2. (Sikiric et al.)

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TB-500: Cell Migration

Sequesters G-actin and promotes cell migration toward injury sites. The fragment is the actin-binding region of thymosin beta-4, not the whole protein. FDA Category 2. WADA prohibited. (Goldstein et al.)

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Fixed 1:1 Ratio

One draw delivers both at the vial's proportion. Neither component can be titrated, paused or withdrawn independently of the other.

Combination: Unvalidated

No published research examines these two peptides together. Whether the effects add, do nothing, or interfere is unknown and untested.

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Co-formulation Stability

The stability of two peptides stored and reconstituted in the same vial has not been validated in published research.

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Route

Subcutaneous injection after reconstitution with bacteriostatic water. The circulated amounts assume that route; no human study establishes it for either peptide.

Research Timeline

1993
BPC First Described
Sikiric and colleagues describe a peptide isolated from human gastric juice and set out the stomach-stress-organoprotection hypothesis. This is the origin of the BPC-157 literature.
2004
Thymosin Beta-4 Cardiac Repair Study
Bock-Marquette et al. publish in Nature showing thymosin beta-4 promotes cardiac cell migration, survival and repair in mice. The study used the full 43-amino-acid protein, not the 7-amino-acid TB-500 fragment sold today.
1993–2020
Preclinical BPC-157 Programme Expands
The Zagreb group publishes extensively on wound healing, tendon and ligament repair, and gastrointestinal protection. The work is overwhelmingly in rodents, and no human trial establishing a subcutaneous schedule follows from it.
2012
TB-500 Detection and Review
Goldstein et al. publish a review of thymosin beta-4 as a regenerative peptide. Separately, Ho et al. publish a doping-control assay for TB-500 in equine urine and plasma — the compound is by then circulating widely enough to require testing for.
2023
FDA Places Both Components in Category 2
The FDA lists BPC-157 and TB-500 among bulk drug substances that may present significant safety risks, prohibiting their compounding for human use. Neither is approved for any therapeutic indication.
2024–2025
First Human BPC-157 Reports
Small human reports appear — an intravenous safety and pharmacokinetics pilot, and an intravesical preliminary report in interstitial cystitis. A systematic review of orthopaedic use concludes the human evidence base remains insufficient. None of this work uses subcutaneous injection or establishes a schedule.
2024–2026
Two-Peptide Repair Blends Commercialised
BPC-157 and TB-500 are widely sold pre-mixed in a single vial under names such as Wolverine. Marketing emphasises combined repair. No published study of the combination exists at the time of writing, and the amounts circulated for it are not traceable to a trial.

Contraindications & Safety Data

There is no safety data on this combination. What follows is drawn from the two component literatures, which are themselves almost entirely preclinical. Interactions between the two peptides are uncharacterised.

ConcernRisk levelRationale
Active cancer or malignancyHIGHBoth components are associated with angiogenesis and cell migration in preclinical models. Both mechanisms could theoretically support tumour growth and vascularisation.
FDA Category 2 classification (both components)HIGH (regulatory)BPC-157 and TB-500 are both listed by the FDA as presenting significant safety risks and are prohibited from compounding for human use.
Pregnancy or breastfeedingHIGHNo reproductive safety data exists for either component or the combination. Standard exclusion for unstudied compounds.
Competitive athletes subject to testingHIGH (sanction)Both components appear on the WADA Prohibited List under S0, banned at all times, in and out of competition. Validated detection assays for TB-500 have existed since 2012.
Drug interactionsUNKNOWNNo interaction study exists for either peptide, in combination or with any medicine. Pharmacokinetic and pharmacodynamic interactions are uncharacterised.
Fixed ratio, no independent titrationMODERATE (practical)A single draw delivers both peptides. Reducing exposure to one necessarily reduces the other, and an adverse response cannot be attributed to a component or managed by adjusting it.
Co-formulation stabilityUNKNOWNDegradation kinetics and possible interactions between two peptides stored together, dry and in solution, have not been validated in published research.
Vial size against reconstituted shelf lifeMODERATE (practical)At the amounts circulated for this blend a 20 mg vial holds forty to eighty daily doses, well beyond the roughly four weeks a reconstituted vial is generally held to keep for under refrigeration.
Human safety data (individual components)LIMITED TO ABSENTNo published human study establishes a subcutaneous amount, schedule or duration for either peptide. The small BPC-157 human reports used other routes; the human thymosin beta-4 work used the full protein rather than the TB-500 fragment.
Human safety data (combination)ABSENTNo published study of any kind examines BPC-157 and TB-500 co-administered, in any model system.
Quality control and vendor variationVARIABLEPurity, sterility and the accuracy of the stated 10 + 10 mg fill vary by supplier. A blend adds a second peptide's assay to what a certificate of analysis has to establish.

Regulatory Status

FDA: Neither component is approved for any therapeutic use. Both are listed as Category 2 bulk drug substances, meaning the agency has identified significant safety risks and prohibited their compounding for human use. The blend has no separate regulatory status of its own.

WADA: Both components fall under S0 (Non-Approved Substances) on the Prohibited List, banned at all times, in and out of competition.

DEA: Neither component is a scheduled substance.

Key distinction: A blend is not evidence of a combination. Pre-mixing two peptides makes them easier to inject together; it does not generate data about what they do together, and it removes the ability to vary them independently. On the evidence available, Wolverine is two under-studied compounds in one vial rather than a studied product.

References (APA 7th Edition)

Sikiric, P., Petek, M., Rucman, R., Seiwerth, S., Grabarevic, Z., Rotkvic, I., ... & Duvnjak, M. (1993). A new gastric juice peptide, BPC: An overview of the stomach-stress-organoprotection hypothesis and beneficial effects of BPC. Journal of Physiology and Pharmacology, 44(6), 601–609.
Sikiric, P., Rucman, R., Turkovic, B., et al. (2018). Novel cytoprotective mediator, stable gastric pentadecapeptide BPC 157: Vascular recruitment and gastrointestinal tract healing. Current Pharmaceutical Design, 24(18), 2002–2030.
Vasireddi, N., Hahamyan, H., Salata, M. J., Karns, M., Calcei, J. G., Voos, J. E., & Apostolakos, J. M. (2025). Emerging use of BPC-157 in orthopaedic sports medicine: A systematic review. Orthopaedic Journal of Sports Medicine.
Lee, Y. K., & Burgess, L. (2025). Intravenous BPC-157 safety and pharmacokinetics in healthy adults: A pilot study. Clinical Pharmacology in Drug Development.
Bock-Marquette, I., Saxena, A., White, M. D., DiMaio, J. M., & Srivastava, D. (2004). Thymosin beta-4 activates integrin-linked kinase and promotes cardiac cell migration, survival and cardiac repair. Nature, 432(7016), 466–472.
Goldstein, A. L., Hannappel, E., Sosne, G., & Kleinman, H. K. (2012). Thymosin beta-4: A multi-functional regenerative peptide. Basic properties and clinical applications. Expert Opinion on Biological Therapy, 12(1), 37–51.
Ho, E. N., Kwok, W., Lau, M., Wong, A. S., Wan, T. S., Lam, K. K., Schiff, P. J., & Stewart, B. D. (2012). Doping control analysis of TB-500 in equine urine and plasma by liquid chromatography–mass spectrometry. Journal of Chromatography B, 900, 78–83.
Rahaman, K. A., Muresan, A. R., Min, H., Son, J., Han, H., Kang, M., & Kwon, O. (2024). Simultaneous quantification of TB-500 and its metabolites in in-vitro experiments and rats by UHPLC-Q-Exactive orbitrap MS/MS and their screening by wound healing activities in-vitro. Journal of Pharmaceutical Analysis.
U.S. Food and Drug Administration. (2023). Certain bulk drug substances for use in compounding that may present significant safety risks. FDA.
World Anti-Doping Agency. (2024). The 2025 World Anti-Doping Code International Standard: Prohibited List. WADA.
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Educational Disclaimer

This profile is for educational and research purposes only. It is not medical advice, and nothing on it is a protocol, a recommendation, or an instruction for use in a person or an animal.

Athena Peptides Education does not prescribe, sell, or recommend any compound. Compounds discussed here are for laboratory research only and are not for human consumption. Always consult a qualified physician before making any decision about your health.